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 3-iodo-1H-indazole YC-1 (2S,3S,4R,5R,6S)-5-(benzyloxy)-6-((5,7-bis(benzyloxy)-2-(4-(benzyloxy)phenyl)-4-oxo-4H-chromen-3-yl)oxy)-2-methyltetrahydro-2H-pyran-3,4-diyl diacetate (2S,3S,4R,5R,6S)-5-(benzyloxy)-6-bromo-2-methyltetrahydro-2H-pyran-3,4-diyl diacetate
 (2S,3S,4R,5R,6S)-5-(benzyloxy)-2-methyl-6-(phenylthio)tetrahydro-2H-pyran-3,4-diyl diacetate (2S,3R,4R,5R,6S)-5-(benzyloxy)-2-methyl-6-(phenylthio)tetrahydro-2H-pyran-3,4-diol (4aS,5S,7S,8R,8aR)-8-(benzyloxy)-2,3-dimethoxy-2,3,5-trimethyl-7-(phenylthio)hexahydro-2H-pyrano[3,4-b][1,4]dioxine (4aS,5S,7S,8R,8aS)-2,3-dimethoxy-2,3,5-trimethyl-7-(phenylthio)hexahydro-2H-pyrano[3,4-b][1,4]dioxin-8-ol
 (2S,3R,4R,5R,6S)-2-methyl-6-(phenylthio)tetrahydro-2H-pyran-3,4,5-triol (2S,3S,4R,5R,6S)-2-methyl-6-(phenylthio)tetrahydro-2H-pyran-3,4,5-triyl triacetate (2S,3R,4R,5S,6S)-6-methyltetrahydro-2H-pyran-2,3,4,5-tetrayl tetraacetate 5,7-bis(benzyloxy)-2-(4-(benzyloxy)phenyl)-3-hydroxy-4H-chromen-4-one
 5,7-bis(benzyloxy)-2-(4-(benzyloxy)phenyl)-4H-chromen-4-one (E)-3-(4-(benzyloxy)phenyl)-1-(2,4-bis(benzyloxy)-6-hydroxyphenyl)prop-2-en-1-one SL-0101 5-cyano-2’-(piperazin-1-yl)-N-(3-(pyrrolidin-1-yl)propyl)-[1,1’-biphenyl]-3-carboxamide
 tert-butyl 4-(3’-cyano-5’-((3-(pyrrolidin-1-yl)propyl)carbamoyl)-[1,1’-biphenyl]-2-yl)piperazine-1-carboxylate 2’-bromo-5-cyano-N-(3-(pyrrolidin-1-yl)propyl)-[1,1’-biphenyl]-3-carboxamide LLY-507 2,2-dimethyl-4-((4-(2-(4-(oxiran-2-ylmethoxy)phenyl)propan-2-yl)phenoxy)methyl)-1,3-dioxolane
 EPI-001 ETC-1002 (ESP 55016),Bempedoic Acid 2-(3-bromophenyl)-N-((3’-(methylsulfonyl)-[1,1’-biphenyl]-4-yl)methyl)ethanamine 3’-(methylsulfonyl)-[1,1’-biphenyl]-4-carboxylic acid
 SR9243 N-(2-oxoindolin-5-yl)-3-(piperidin-1-yl)propanamide 5-aminoindolin-2-one DEL-22379,HY-18932
 MCB-613 (R)-tert-butyl 3-((6-(dibenzylamino)-5-nitropyrimidin-4-yl)amino)piperidine-1-carboxylate N,N-dibenzyl-6-chloro-5-nitropyrimidin-4-amine ethyl 4-((1,5-dimethyl-1H-pyrazol-3-yl)amino)-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxylate
 3-iodo-1,5-dimethyl-1H-pyrazole 1,5-dimethyl-1H-pyrazol-3-amine ethyl 4-(4-cyano-1-methyl-1H-imidazol-5-yl)-1-ethyl-1H-pyrrole-2-carboxylate 5-bromo-1-methyl-1H-imidazole-4-carbonitrile
 1-methyl-1H-imidazole-4-carbonitrile (E)-3-(pyrrolidin-1-yl)-2-((E)-(pyrrolidin-1-ylmethylene)amino)acrylonitrile ethyl 4-bromo-1-ethyl-1H-pyrrole-2-carboxylate ethyl 4-bromo-1H-pyrrole-2-carboxylate
 1-(4-bromo-1H-pyrrol-2-yl)-2,2,2-trichloroethanone BMS-911543 1-(6-methylpyridin-2-yl)-2-(1,5-naphthyridin-2-yl)ethanone 2-methyl-1,5-naphthyridine
 Alk5i 1-(((S)-3-(diethylamino)-2-hydroxypropyl)amino)-4-(((S)-oxiran-2-ylmethyl)amino)anthracene-9,10-dione sodium 4-methylbenzenesulfonate (E)-3-tosylacrylonitrile
 (Z)-3-(((4-((dimethylamino)methyl)phenyl)amino)(phenyl)methylene)-6-iodoindolin-2-one (E)-6-iodo-3-(phenyl((trimethylsilyl)oxy)methylene)-2-((trimethylsilyl)oxy)-3H-indole (S)-tert-butyl 4-((((9H-fluoren-9-yl)methoxy)carbonyl)amino)-5-(((S)-1-(allyloxy)-3-methyl-1-oxobutan-2-yl)amino)-5-oxopentanoate (S)-allyl 2-amino-3-methylbutanoate
 Ac-DEVD-CHO (E)-methyl 4-(3-(dimethylamino)-2-methylacryloyl)-1-tosyl-1H-pyrrole-2-carboxylate methyl 4-propionyl-1-tosyl-1H-pyrrole-2-carboxylate methyl 4-propionyl-1H-pyrrole-2-carboxylate
 1-(5-(2,2,2-trichloroacetyl)-1H-pyrrol-3-yl)propan-1-one VX-11e 1-(3-fluoro-2-(trifluoromethyl)isonicotinoyl)piperidin-4-one piperidin-4-one hydrochloride
 tert-butyl 3-(cyanomethyl)-3-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl)azetidine-1-carboxylate tert-butyl 3-(cyanomethylene)azetidine-1-carboxylate tert-butyl 3-oxoazetidine-1-carboxylate tert-butyl 3-hydroxyazetidine-1-carboxylate
 INCB39110 (1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazol-5-yl)boronic acid 1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazole 8-ethyl-4-methyl-2-(methylthio)-6-(1H-pyrazol-5-yl)pyrido[2,3-d]pyrimidin-7(8H)-one
 8-ethyl-4-methyl-2-(methylthio)pyrido[2,3-d]pyrimidin-7(8H)-one (E)-ethyl 3-(4-(ethylamino)-6-methyl-2-(methylthio)pyrimidin-5-yl)acrylate N-ethyl-5-iodo-6-methyl-2-(methylthio)pyrimidin-4-amine N-ethyl-6-methyl-2-(methylthio)pyrimidin-4-amine
 4-chloro-6-methyl-2-(methylthio)pyrimidine 6-methyl-2-(methylthio)pyrimidin-4(3H)-one Voxtalisib (XL765, SAR245409) thiazol-5-ylboronic acid
 2-(trimethylsilyl)thiazole 6-(4-bromo-2-chlorophenyl)-8-ethyl-2-((4-(4-methylpiperazin-1-yl)phenyl)amino)pyrido[2,3-d]pyrimidin-7(8H)-one 6-(4-bromo-2-chlorophenyl)-2-chloro-8-ethylpyrido[2,3-d]pyrimidin-7(8H)-one methyl 2-(4-bromo-2-chlorophenyl)acetate
 2-(4-bromo-2-chlorophenyl)acetonitrile 4-bromo-1-(bromomethyl)-2-chlorobenzene 2-chloro-4-(ethylamino)pyrimidine-5-carbaldehyde (2-chloro-4-(ethylamino)pyrimidin-5-yl)methanol
 ethyl 2-chloro-4-(ethylamino)pyrimidine-5-carboxylate FRAX597 ethyl 3-(3-(tert-butylthio)-1-(4-(6-ethoxypyridin-3-yl)benzyl)-5-((5-methylpyridin-2-yl)methoxy)-1H-indol-2-yl)-2,2-dimethylpropanoate 2-ethoxy-5-(4-((1-(4-((5-methylpyridin-2-yl)methoxy)phenyl)hydrazinyl)methyl)phenyl)pyridine
 4-((5-methylpyridin-2-yl)methoxy)aniline 5-(4-(bromomethyl)phenyl)-2-ethoxypyridine (4-(6-ethoxypyridin-3-yl)phenyl)methanol GSK2190915 (AM803)
 2,3,5-trifluoro-N-(3-fluoro-4-iodophenyl)-6-nitroaniline (S)-1-((2,2-dimethyl-1,3-dioxolan-4-yl)methyl)cyclopropane-1-sulfonyl chloride (S)-butyl 1-(3-((tert-butyldimethylsilyl)oxy)-2-hydroxypropyl)cyclopropane-1-sulfonate O-(2-(vinyloxy)ethyl)hydroxylamine
 2-(2-(vinyloxy)ethoxy)isoindoline-1,3-dione 5-((4-bromo-2-fluorophenyl)amino)-4-fluoro-1-methyl-N-(2-(vinyloxy)ethoxy)-1H-benzo[d]imidazole-6-carboxamide 5-((4-bromo-2-fluorophenyl)amino)-4-fluoro-1-methyl-1H-benzo[d]imidazole-6-carboxylic acid methyl 6-((4-bromo-2-fluorophenyl)amino)-7-fluoro-1H-benzo[d]imidazole-5-carboxylate
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